19. Drug Effects, Toxicities, and Poisonings in Children

Accidental pediatric ingestions and therapeutic drug toxicities represent critical medical emergencies requiring rapid recognition of toxidromes and toxic electrocardiographic patterns.


1. Common Cardiotoxic Agents & Electrocardiographic Hallmarks

Drug ClassMechanism of CardiotoxicityClassical 12-Lead Electrocardiographic HallmarksSpecific Antidote / Treatment
Tricyclic Antidepressants (TCA)Fast $Na^+$ channel blockade ($I_{Na}$) + Anticholinergic effect.Terminal R wave in aVR $>3\text{ mm}$, $R/S$ in aVR $>0.7$, prolonged QRS ($>100\text{ ms}$), sinus tachycardia, prolonged $QTc$.IV Sodium Bicarbonate ($8.4\%$): $1-2\text{ mEq/kg}$ IV push to alkalinize serum to pH $7.45-7.55$.
Digoxin (Cardiac Glycosides)$Na^+/K^+$ ATPase inhibition $\to$ intracellular $Ca^{2+}$ overload.Effect: "Scooped" sagging ST depression (reverse tick mark), short QTc.
Toxicity: Ventricular bigeminy, bidirectional VT, high-grade AV block.
Digoxin Immune Fab (DigiFab); IV Magnesium Sulfate; avoid electrical cardioversion if possible.
Beta-Adrenergic BlockersCompetitive antagonism of $\beta_1$ and $\beta_2$ receptors.Severe sinus bradycardia, first/second/third-degree AV block, junctional escape rhythm, prolonged QRS (propranolol).High-Dose Insulin Euglycemia (HIE) + IV Glucagon ($50-100\ \mu\text{g/kg}$) + Calcium Gluconate.
Calcium Channel Blockers (CCB)L-type $Ca^{2+}$ channel blockade.Sinus arrest, complete AV block, PR prolongation, refractory cardiogenic shock with hyperglycemia.High-Dose Insulin Euglycemia (HIE) + IV Calcium Chloride $10\%$ + Lipid Emulsion Therapy ($20\%$).

2. Emergency Management Protocols

ACUTE TRICYCLIC ANTIDEPRESSANT (TCA) OVERDOSE │ ┌──────────────────────┴──────────────────────┐ QRS Duration > 100 ms QRS Duration > 160 ms (Risk of Generalized Seizures) (High Risk of Ventricular Arrhythmias) │ │ IV Sodium Bicarbonate IV Sodium Bicarbonate (1-2 mEq/kg bolus -> Continuous (Immediate bolus + Infusion; Infusion to target pH 7.45-7.55) Avoid Physostigmine / Class IA)


3. Clinical Pearls & Diagnostic Traps

Red Flag Warning: Never administer Class IA (Procainamide, Quinidine) or Class IC (Flecainide) antiarrhythmics to treat wide-complex tachycardias caused by TCA or sodium channel blocker poisoning. They will compound myocardial sodium channel blockade and precipitate fatal asystole.